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GP 1a
CAS No. 511532-96-0
GP 1a( —— )
Catalog No. M35265 CAS No. 511532-96-0
GP 1a is a potent agonist of cannabinoid receptor 2 (CB2) (EC50=7.1), as shown in cAMP, GTPγS and β-arrestin recruitment assays.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 78 | Get Quote |
|
| 5MG | 107 | Get Quote |
|
| 10MG | 169 | Get Quote |
|
| 25MG | 330 | Get Quote |
|
| 50MG | 490 | Get Quote |
|
| 100MG | 683 | Get Quote |
|
| 500MG | 1377 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameGP 1a
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NoteResearch use only, not for human use.
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Brief DescriptionGP 1a is a potent agonist of cannabinoid receptor 2 (CB2) (EC50=7.1), as shown in cAMP, GTPγS and β-arrestin recruitment assays.
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DescriptionGP1a is a potent agonist of cannabinoid receptor 2 (CB2). Gp1a is beneficial to skin wound healing. GP1a inhibits inflammation and fibrogenesis while promoting re-epithelialization.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCannabinoid Receptor | PERK
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Research Area——
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Indication——
Chemical Information
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CAS Number511532-96-0
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Formula Weight441.35
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Molecular FormulaC23H22Cl2N4O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (283.22 mM; Ultrasonic )
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SMILESC(NN1CCCCC1)(=O)C=2C3=C(N(N2)C4=C(Cl)C=C(Cl)C=C4)C=5C(C3)=CC(C)=CC5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhao C, et al. An enzyme-responsive Gp1a-hydrogel for skin wound healing. J Biomater Appl. 2021;36(4):714-721.?
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